US Patent:
20130237573, Sep 12, 2013
Inventors:
Bruce Anthony Dressman - Indianapolis IN, US
Mark Donald Chappell - Indianapolis IN, US
Adam Michael Fivush - Fishers IN, US
Charles Howard Mitch - Columbus IN, US
Paul Leslie Ornstein - Carmel IN, US
Eric George Tromiczak - Indianapolis IN, US
Tatiana Natali Vetman - Greenwood IN, US
Assignee:
ELI LILLY AND COMPANY - Indianapolis IN
International Classification:
C07D 277/36
A61K 31/4196
A61K 31/4164
A61K 31/27
A61K 45/06
A61K 31/265
A61K 31/216
A61K 31/196
C07D 249/12
C07D 235/00
C07C 69/96
C07C 271/24
C07C 69/757
C07C 62/34
A61K 31/135
A61K 31/426
US Classification:
514369, 514384, 514398, 514479, 514480, 514512, 514530, 514570, 548187, 5482642, 5483251, 558267, 560 27, 560 45, 562455
Abstract:
A mGlu2/3 receptor antagonist of the formula:its uses, and methods for its preparation are described.