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Gerald P Lelais

from San Diego, CA
Age ~48

Gerald Lelais Phones & Addresses

  • 3965 Caminito Del Mar Surf, San Diego, CA 92130 (858) 847-0571
  • Pasadena, CA

Work

Company: Gnf Jan 2010 Position: Research investigator ii

Education

Degree: Postdoctoral Research Fellow School / High School: California Institute of Technology 2004 to 2006 Specialities: Chemistry

Skills

Organic Chemistry • Drug Discovery • Medicinal Chemistry • Lead Change • Drug Design • Research • Gpcrs • Kinases

Languages

Italian • French • German • English

Industries

Pharmaceuticals

Resumes

Resumes

Gerald Lelais Photo 1

Associate Director

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Location:
1619 Stanford St, Santa Monica, CA 90404
Industry:
Pharmaceuticals
Work:
GNF since Jan 2010
Research Investigator II

GNF Oct 2006 - Dec 2009
Research Investigator I
Education:
California Institute of Technology 2004 - 2006
Postdoctoral Research Fellow, Chemistry
Eidgenössische Technische Hochschule Zürich 2000 - 2004
Ph.D., Chemistry
Eidgenössische Technische Hochschule Zürich 1995 - 2000
B.S., Chemistry
Skills:
Organic Chemistry
Drug Discovery
Medicinal Chemistry
Lead Change
Drug Design
Research
Gpcrs
Kinases
Languages:
Italian
French
German
English

Business Records

Name / Title
Company / Classification
Phones & Addresses
Gerald Lelais
ManagingPrincipal
Silver Treasure LLC
Online Business Selling Sterling Silver · Business Services at Non-Commercial Site
13335 Tiverton Rd, San Diego, CA 92130
3965 Caminito Del Mar Surf, San Diego, CA 92130

Publications

Us Patents

4-Phenoxymethylpiperidines As Modulators Of Gpr119 Activity

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US Patent:
8334288, Dec 18, 2012
Filed:
Jul 9, 2009
Appl. No.:
13/003558
Inventors:
Robert Epple - San Diego CA, US
Gerald Lelais - San Diego CA, US
Victor Nikulin - Carlsbad CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/496
C07D 241/02
C07D 401/00
US Classification:
51425211, 51425301, 544357, 544360, 544405
Abstract:
The present invention provides compounds of Formula I, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent; diseases or disorders associated with the activity of GPR119.

Compounds And Methods For Modulating G Protein-Coupled Receptors

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US Patent:
8394841, Mar 12, 2013
Filed:
Jan 8, 2008
Appl. No.:
12/527849
Inventors:
Robert Epple - San Diego CA, US
Mihai Azimioara - San Diego CA, US
Christopher Cow - San Diego CA, US
Ross Russo - Encinitas CA, US
Victor Nikulin - San Diego CA, US
Gerald Lelais - San Diego CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/426
A61K 31/421
C07D 277/20
C07D 263/30
US Classification:
514365, 435375, 514374, 548202, 548235
Abstract:
The invention provides compounds and pharmaceutical compositions thereof, which are useful for modulating G protein-coupled receptor 120 (GPR120), and methods for using such compounds to treat, ameliorate or prevent a condition associated with abnormal or deregulated GPR120.

Compounds And Compositions As Modulators Of Gpr119 Activity

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US Patent:
8575168, Nov 5, 2013
Filed:
Oct 1, 2010
Appl. No.:
12/896735
Inventors:
Mihai Azimioara - La Jolla CA, US
Christopher Cow - Poway CA, US
Robert Epple - San Diego CA, US
Gerald Lelais - San Diego CA, US
John Mecom - San Diego CA, US
Victor Nikulin - Carlsbad CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/497
A61K 31/445
C07D 239/42
C07D 239/00
C07D 241/00
C07D 401/00
C07D 405/00
US Classification:
5142521, 51425212, 51425213, 514256, 514315, 514316, 544242, 544336, 544360, 546187
Abstract:
The invention provides compounds, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent diseases or disorders associated with the activity of GPR119.

Compounds And Compositions As Modulators Of Gpr119 Activity

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US Patent:
20090270409, Oct 29, 2009
Filed:
Sep 4, 2008
Appl. No.:
12/204600
Inventors:
Phillip B. Alper - San Diego CA, US
Mihai Azimioara - La Jolla CA, US
Christopher Cow - San Diego CA, US
Robert Epple - San Diego CA, US
Songchun Jiang - San Diego CA, US
Gerald Lelais - San Diego CA, US
Pierre-Yves Michellys - San Marcos CA, US
Daniel Mutnick - San Diego CA, US
Victor Nikulin - Carlsbad CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/497
C07D 401/02
C07D 409/14
C07D 241/04
US Classification:
51425211, 544360, 544364, 544357, 51425313, 51425309
Abstract:
The invention provides compounds, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent diseases or disorders associated with the activity of GPR119.

Compounds And Compositions As Modulators Of Gpr119 Activity

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US Patent:
20100022515, Jan 28, 2010
Filed:
Jan 22, 2008
Appl. No.:
12/525289
Inventors:
Phillip B. Alper - San Diego CA, US
Mihai D. Azimioara - La Jolla CA, US
Christopher Cow - San Diego CA, US
Robert Epple - San Diego CA, US
Songchun Jiang - San Diego CA, US
Gerald Lelais - San Diego CA, US
Pierre-Yves Michellys - San Marcos CA, US
Truc Ngoc Nguyen - San Diego CA, US
Baogen Wu - San Diego CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/55
C07D 401/14
A61K 31/4709
A61K 31/5377
A61K 31/497
C07D 413/14
C07D 401/12
US Classification:
51421301, 546153, 514312, 5142352, 51425307, 544363, 544128, 540593
Abstract:
The invention provides compounds, pharmaceutical compositions comprising compound of following formula (I), and methods of using such compounds to treat or prevent diseases or disorders associated with the activity of GPR119 (G protein-coupled receptor 119) such as obesity, diabetes and hyperlipidemia.

Thiazole Derivatives As Modulators Of G Protein-Coupled Receptors

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US Patent:
20100022592, Jan 28, 2010
Filed:
Jan 7, 2008
Appl. No.:
12/527826
Inventors:
Robert Epple - San Diego CA, US
Mihai Azimioara - San Diego CA, US
Christopher Cow - San Diego CA, US
Ross Russo - Encinitas CA, US
Victor Nikulin - Carlsbad CA, US
Gerald Lelais - San Diego CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/427
C07D 417/10
C07D 417/14
C12N 5/00
A61K 31/454
A61K 31/4439
A61P 3/10
US Classification:
514326, 548202, 5462704, 546209, 435375, 514342, 514365
Abstract:
The invention provides compounds of formula (IA) or (IB) and pharmaceutical compositions thereof, which are useful for modulating G protein-coupled receptor 120 (GPR120), and methods for using such compounds to treat, ameliorate or prevent a condition associated with abnormal or deregulated GPR120.

Compounds And Compositions As Modulators Of Gpr119 Activity

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US Patent:
20100120807, May 13, 2010
Filed:
Mar 5, 2008
Appl. No.:
12/529694
Inventors:
Phillip B. Alper - San Diego CA, US
Gerald Lelais - San Diego CA, US
Robert Epple - SAn Diego CA, US
Daniel Mutnick - San Diego CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/454
C07D 413/04
C07D 401/14
C07D 413/14
A61K 31/506
A61P 3/04
A61P 3/10
A61P 9/00
A61P 9/10
A61P 19/00
A61P 3/06
A61P 7/00
A61P 19/02
A61P 19/10
A61P 9/12
A61P 27/02
A61P 27/12
A61P 13/12
A61P 25/00
A61P 3/00
A61P 15/00
A61P 7/02
A61P 3/08
A61P 5/48
A61P 15/10
A61P 17/00
A61P 19/04
A61P 17/02
A61P 1/04
US Classification:
514275, 546209, 546210, 544331, 514326
Abstract:
The invention provides compounds, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent diseases or disorders associated with the activity of GPR119.

Compounds And Compositions As Modulators Of Gpr119 Activity

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US Patent:
20110190263, Aug 4, 2011
Filed:
Feb 20, 2009
Appl. No.:
12/918803
Inventors:
Mihai Azimioara - La Jolla CA, US
Christopher Cow - Poway CA, US
Robert Epple - San Diego CA, US
Songchun Jiang - San Diego CA, US
Gerald Lelais - San Diego CA, US
Baogen Wu - San Diego CA, US
Daniel Mutnick - San Diego CA, US
Assignee:
IRM LLC - Hamilton
International Classification:
A61K 31/519
C12N 5/02
C07D 471/04
A61K 31/506
A61P 3/04
A61P 3/10
A61P 3/06
A61P 9/00
A61P 19/02
A61P 19/10
A61P 9/02
A61P 13/12
A61P 17/00
A61P 1/00
US Classification:
51421021, 435375, 544279, 514275, 544297
Abstract:
The invention provides compounds of Formula (I): pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent diseases or disorders associated with the activity of GPR119.
Gerald P Lelais from San Diego, CA, age ~48 Get Report